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Synthesis, structure-activity relationships, and docking studies of N-phenylarylformamide derivatives (PAFAs) as non-nucleoside HIV reverse transcriptase inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2012, 卷号: 58, 期号: X, 页码: 504-512
作者:  Ma XD;  He QQ;  Zhang X;  Yang SQ;  Yang LM;  Gu SX;  Zheng YT;  Chen FE*;  Dai HF*;  rfchen@fudan.edu.cn
Adobe PDF(825Kb)  |  收藏  |  浏览/下载:135/3  |  提交时间:2013/03/08
Anti-hiv Activity  Nnrtis  Benzophenone Derivatives  N-phenylarylformamide  Structure-activity Relationship  
Synthesis and biological evaluation of novel dihydro-aryl/alkylsulfanyl-cyclohexylmethyl-oxopyrimidines (S-DACOs) as high active anti-HIV agents 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 卷号: 21, 期号: 2, 页码: 694-697
作者:  He YP*;  Long J;  Zhang SS;  Li C;  Lai CC;  Zhang CS;  Li DX;  Zhang DH;  Wang H;  Cai QQ;  Zheng YT*;  yphe@ynu.edu.cn;  zhengyt@mail.kiz.ac.cn
Adobe PDF(395Kb)  |  收藏  |  浏览/下载:1658/7  |  提交时间:2011/03/15
Nnrtis  S-dabos  S-dacos  Anti Hiv-1 Activity  
Synthesis and biological evaluation of (+/-)-benzhydrol derivatives as potent non-nucleoside HIV-1 reverse transcriptase inhibitors 期刊论文
Bioorganic & Medicinal Chemistry, 2011, 卷号: 19, 期号: 16, 页码: 4704-4709
作者:  Ma XD;  Zhang X;  Yang SQ;  Dai HF;  Yang LM;  Gu SX;  Zheng YT;  He QQ;  Chen FE*;  rfchen@fudan.edu.cn
Adobe PDF(595Kb)  |  收藏  |  浏览/下载:113/4  |  提交时间:2011/08/18
Hiv  Nnrtis  Benzophenone Derivatives  Benzhydrol  Sar  
Synthesis and biological activity of naphthyl-substituted (B-ring) benzophenone derivatives as novel non-nucleoside HIV-1 reverse transcriptase inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2011, 卷号: 19, 期号: 15, 页码: 4601-4607
作者:  Ma XD;  Zhang X;  Dai HF;  Yang SQ;  Yang LM;  Gu SX;  Zheng YT;  He QQ;  Chen FE*;  rfchen@fudan.edu.cn
Adobe PDF(461Kb)  |  收藏  |  浏览/下载:125/3  |  提交时间:2011/08/09
Hiv  Nnrtis  Benzophenone Derivatives  Naphthyl  Sar  
Synthesis and biological evaluation of naphthyl phenyl ethers (NPEs) as novel nonnucleoside HIV-1 reverse transcriptase inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 卷号: 19, 期号: 14, 页码: 4220-4226
作者:  Gu SX;  Zhang X;  Zheng YT;  Yang SQ;  Chen FE*;  He QQ;  Yang LM;  Ma XD;  rfchen@fudan.edu.cn
Adobe PDF(416Kb)  |  收藏  |  浏览/下载:55/1  |  提交时间:2016/08/30
Hiv-1 Reverse Transcriptase  Nnrtis  Npes  Sar  Anti-hiv Activity  
Synthesis and biological evaluation of (+/-)-benzhydrol derivatives as potent non-nucleoside HIV-1 reverse transcriptase inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2011, 卷号: 19, 期号: 16, 页码: 4704-4709
作者:  Ma XD;  Zhang X;  Yang SQ;  Dai HF;  Yang LM;  Gu SX;  Zheng YT;  He QQ;  Chen FE*;  rfchen@fudan.edu.cn
Adobe PDF(595Kb)  |  收藏  |  浏览/下载:1629/3  |  提交时间:2011/08/26
Hiv  Nnrtis  Benzophenone Derivatives  Benzhydrol  Sar  
The anti-HIV activity of three 2-alkylsulfanyl-6-benzyl-3, 4- dihydropyrimidin-4 (3H)-one derivatives acting as non-nucleoside reverse transcriptase inhibitor in vitro 期刊论文
药学学报, 2010, 卷号: 45, 期号: 2, 页码: 228-234
作者:  Long J;  Zhang DH;  Zhang GH;  Rao ZK;  Wang YH;  Tam SC;  He YP*;  Zheng YT*;  yphe@ynu.edu.cn;  zhengyt@mail.kiz.ac.cn
Adobe PDF(850Kb)  |  收藏  |  浏览/下载:120/4  |  提交时间:2010/08/19
Aids  Hiv-1  Reverse Transcriptase  Nnrtis  S-dabos  Anti-hiv Activity  
Synthesis and anti-HIV-1 activity of S-dihydro(alkyloxy)benzyloxypyrimidine derivatives 期刊论文
MONATSHEFTE FUR CHEMIE, 2008, 卷号: 139, 期号: 8, 页码: 967-974
作者:  Rao ZK;  Long J;  Zhang SS;  He M;  Ou LC;  Zheng YT*;  He YP*;  Li C;  zhengyt@mail.kiz.ac.cn;  yphe@ynu.edu.cn
Adobe PDF(309Kb)  |  收藏  |  浏览/下载:86/4  |  提交时间:2010/08/24
Nnrtis  S-dabos  Antiviral Activity  Hiv-1  
Synthesis and biological evaluation of N-acetyl-beta-aryl-1,2-didehydroethylamines as new HIV-1 RT inhibitors in vitro 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2007, 卷号: 17, 期号: 16, 页码: 4476-4480
作者:  Cheng P;  Jiang ZY;  Wang RR;  Zhang XM;  Wang Q;  Zheng YT*;  Zhou J;  Chen JJ*;  chenjj@mail.kib.ac.cn
Adobe PDF(148Kb)  |  收藏  |  浏览/下载:93/4  |  提交时间:2010/08/24
Beta-aryl-nitroolefin  N-acetyl-beta-aryl-1  Nnrtis  2-didehydroethylamine  Anti-hiv-1 Rt Activity