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Synthesis and biological evaluation of 5-fluoroquinolone-3-carboxylic acids as potential HIV-1 integrase inhibitors 期刊论文
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2013, 卷号: 28, 期号: 4, 页码: 671-676
作者:  He QQ;  Zhang X;  Yang LM;  Zheng YT;  Chen F*;  rfchen@fudan.edu.cn
Adobe PDF(782Kb)  |  收藏  |  浏览/下载:100/3  |  提交时间:2013/08/27
Hiv-1 Integrase Inhibitor  5-fluoroquinolone-3-carboxylic Acids  Anti-hiv Activity  Metal Chelating  Structure-activity Relationship  
New 23-Spirocholestane Derivatives from Ypsilandra thibetica 期刊论文
PLANTA MEDICA, 2013, 卷号: 79, 期号: 12, 页码: 1063-1067
作者:  Xie BB;  Chen CX;  Guo YH;  Li YY;  Liu YJ;  Ni W;  Yang LM;  Gong NB;  Zheng YT;  Wang RR;  Lu Y;  Liu HY*;  haiyangliu@mail.kib.ac.cn
Adobe PDF(152Kb)  |  收藏  |  浏览/下载:110/2  |  提交时间:2014/10/20
Ypsilandra Thibetica  23-spirocholestane Glycosides  Anti-hiv-1 Activity  Liliaceae  
New Triterpenoids from the Fruits of Schisandra wilsoniana and Their Biological Activities 期刊论文
BULLETIN OF THE KOREAN CHEMICAL SOCIETY, 2013, 卷号: 34, 期号: 3, 页码: 827-830
作者:  Gao XM;  Li YQ;  Shu LD;  Shen YQ;  Yang LY;  Yang LM;  Zheng YT;  Sun HD;  Xiao WL*;  Hu QF*;  xwl@mail.kib.ac.cn;  huqiufena@yahoo.com
Adobe PDF(210Kb)  |  收藏  |  浏览/下载:105/2  |  提交时间:2014/10/17
Schisandra Wilsoniana  Nortriterpenoid  Anti-hiv-1 Activity  Cytotoxicity  
Synthesis and biological evaluation of novel dihydro-aryl/alkylsulfanyl-cyclohexylmethyl-oxopyrimidines (S-DACOs) as high active anti-HIV agents 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 卷号: 21, 期号: 2, 页码: 694-697
作者:  He YP*;  Long J;  Zhang SS;  Li C;  Lai CC;  Zhang CS;  Li DX;  Zhang DH;  Wang H;  Cai QQ;  Zheng YT*;  yphe@ynu.edu.cn;  zhengyt@mail.kiz.ac.cn
Adobe PDF(395Kb)  |  收藏  |  浏览/下载:1658/7  |  提交时间:2011/03/15
Nnrtis  S-dabos  S-dacos  Anti Hiv-1 Activity  
Synthesis and biological evaluation of naphthyl phenyl ethers (NPEs) as novel nonnucleoside HIV-1 reverse transcriptase inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 卷号: 19, 期号: 14, 页码: 4220-4226
作者:  Gu SX;  Zhang X;  Zheng YT;  Yang SQ;  Chen FE*;  He QQ;  Yang LM;  Ma XD;  rfchen@fudan.edu.cn
Adobe PDF(416Kb)  |  收藏  |  浏览/下载:55/1  |  提交时间:2016/08/30
Hiv-1 Reverse Transcriptase  Nnrtis  Npes  Sar  Anti-hiv Activity  
Anti-HIV-1 Activity of Lignans from the Fruits of Schisandra rubriflora 期刊论文
ARCHIVES OF PHARMACAL RESEARCH, 2010, 卷号: 33, 期号: 5, 页码: 697-701
作者:  Xiao WL;  Wang RR;  Zhao W;  Tian RR;  Shang SZ;  Yang LM;  Yang JH;  Pu JX;  Zheng YT;  Sun HD*;  hdsun@mail.kib.ac.cn
Adobe PDF(352Kb)  |  收藏  |  浏览/下载:295/4  |  提交时间:2010/08/24
Schisandra Rubriflora  Lignan  Nmr  Cd Spectrum  Anti-hiv-1 Activity  
The anti-HIV activity of three 2-alkylsulfanyl-6-benzyl-3, 4- dihydropyrimidin-4 (3H)-one derivatives acting as non-nucleoside reverse transcriptase inhibitor in vitro 期刊论文
药学学报, 2010, 卷号: 45, 期号: 2, 页码: 228-234
作者:  Long J;  Zhang DH;  Zhang GH;  Rao ZK;  Wang YH;  Tam SC;  He YP*;  Zheng YT*;  yphe@ynu.edu.cn;  zhengyt@mail.kiz.ac.cn
Adobe PDF(850Kb)  |  收藏  |  浏览/下载:120/4  |  提交时间:2010/08/19
Aids  Hiv-1  Reverse Transcriptase  Nnrtis  S-dabos  Anti-hiv Activity  
Anti-HIV Activities of the Compounds Isolated from Polygonum cuspidatum and Polygonum multiflorum 期刊论文
PLANTA MEDICA, 2010, 卷号: 76, 期号: 9, 页码: 889-892
作者:  Lin HW;  Sun MX;  Wang YH;  Yang LM;  Yang YR;  Huang N;  Xuan LJ;  Xu YM;  Bai DL;  Zheng YT*;  Xiao K*;  zhengyt@mail.kiz.ac.cn;  kaixiaocn@gmail.com
Adobe PDF(123Kb)  |  收藏  |  浏览/下载:326/5  |  提交时间:2010/08/24
Polygonum Cuspidatum  Polygonum Multiflorum  Polygonaceae  Chemical Components  Anti-hiv-1 Activity  
Water-soluble Phenolic Compounds and Their Anti-HIV-1 Activities from the Leaves of Cyclocarya paliurus 期刊论文
JOURNAL OF FOOD AND DRUG ANALYSIS, 2010, 卷号: 18, 期号: 6, 页码: 398-404
作者:  Zhang JA;  Huang N;  Yang LM;  Zheng YT*;  Xiao K*;  Lu JC;  Li X;  Wang YH;  zhengyt@mail.kiz.ac.cn;  kaixiaocn@gmail.com
Adobe PDF(295Kb)  |  收藏  |  浏览/下载:64/2  |  提交时间:2016/09/13
Cyclocarya Paliurus  Phenolics  Flavonol Glucuronides  Anti-hiv-1 Activity  Juglandaceae  
Dibenzocyclooctadiene lignans from the fruits of Schisandra wilsoniana and their anti-HIV-1 activities 期刊论文
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2010, 卷号: 12, 期号: 6, 页码: 470-476
作者:  Yang GY;  Li YK;  Wang RR;  Xiao WL*;  Yang LM;  Pu JX;  Zheng YT;  Sun HD*;  xwl@mail.kib.ac.cn
Adobe PDF(141Kb)  |  收藏  |  浏览/下载:121/2  |  提交时间:2010/08/24
Schisandra Wilsoniana  Fruits  Dibenzocyclooctadiene Lignans  Anti-hiv-1 Activity