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Design, synthesis and anti-HIV-1 evaluation of hydrazide-based peptidomimetics as selective gelatinase inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 9, 页码: 2125-2136
作者:  Yang L;  Wang P;  Pang W;  Li YG;  Shen YM;  Zheng YT*;  Li X*;  Wu JF;  Yang LM;  Wang RR;  zhengyt@mail.kiz.ac.cn;  tjulx2004@sdu.edu.cn
Adobe PDF(3521Kb)  |  收藏  |  浏览/下载:121/4  |  提交时间:2016/04/05
Hydrazide Derivatives  Quinoxalinone  Selective Gelatinase Inhibitors  Peptidomimetics  Anti-hiv Activity  
Identification of the novel N-phenylbenzenesulfonamide derivatives as potent HIV inhibitors 期刊论文
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 2, 页码: 243-247
作者:  Sun YM;  Lu CL;  Wang CY;  Wang RR;  Liu KX;  Yang LM;  Zhen YH;  Zhang HL;  Wang C;  Zheng YT*;  Ma XD*;  zhengyt@mail.kiz.ac.cn;  xiaodong.ma@139.com
Adobe PDF(657Kb)  |  收藏  |  浏览/下载:130/4  |  提交时间:2015/04/24
Benzophenone  N-phenylbenzenesulfonamide  Structure Modification  Anti-hiv Activity  
Synthesis and biological evaluation of 5-fluoroquinolone-3-carboxylic acids as potential HIV-1 integrase inhibitors 期刊论文
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2013, 卷号: 28, 期号: 4, 页码: 671-676
作者:  He QQ;  Zhang X;  Yang LM;  Zheng YT;  Chen F*;  rfchen@fudan.edu.cn
Adobe PDF(782Kb)  |  收藏  |  浏览/下载:100/3  |  提交时间:2013/08/27
Hiv-1 Integrase Inhibitor  5-fluoroquinolone-3-carboxylic Acids  Anti-hiv Activity  Metal Chelating  Structure-activity Relationship  
New 23-Spirocholestane Derivatives from Ypsilandra thibetica 期刊论文
PLANTA MEDICA, 2013, 卷号: 79, 期号: 12, 页码: 1063-1067
作者:  Xie BB;  Chen CX;  Guo YH;  Li YY;  Liu YJ;  Ni W;  Yang LM;  Gong NB;  Zheng YT;  Wang RR;  Lu Y;  Liu HY*;  haiyangliu@mail.kib.ac.cn
Adobe PDF(152Kb)  |  收藏  |  浏览/下载:110/2  |  提交时间:2014/10/20
Ypsilandra Thibetica  23-spirocholestane Glycosides  Anti-hiv-1 Activity  Liliaceae  
New Triterpenoids from the Fruits of Schisandra wilsoniana and Their Biological Activities 期刊论文
BULLETIN OF THE KOREAN CHEMICAL SOCIETY, 2013, 卷号: 34, 期号: 3, 页码: 827-830
作者:  Gao XM;  Li YQ;  Shu LD;  Shen YQ;  Yang LY;  Yang LM;  Zheng YT;  Sun HD;  Xiao WL*;  Hu QF*;  xwl@mail.kib.ac.cn;  huqiufena@yahoo.com
Adobe PDF(210Kb)  |  收藏  |  浏览/下载:105/2  |  提交时间:2014/10/17
Schisandra Wilsoniana  Nortriterpenoid  Anti-hiv-1 Activity  Cytotoxicity  
Synthesis, structure-activity relationships, and docking studies of N-phenylarylformamide derivatives (PAFAs) as non-nucleoside HIV reverse transcriptase inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2012, 卷号: 58, 期号: X, 页码: 504-512
作者:  Ma XD;  He QQ;  Zhang X;  Yang SQ;  Yang LM;  Gu SX;  Zheng YT;  Chen FE*;  Dai HF*;  rfchen@fudan.edu.cn
Adobe PDF(825Kb)  |  收藏  |  浏览/下载:135/3  |  提交时间:2013/03/08
Anti-hiv Activity  Nnrtis  Benzophenone Derivatives  N-phenylarylformamide  Structure-activity Relationship  
Phenols with Anti-HIV Activity from Daphne acutiloba 期刊论文
PLANTA MEDICA, 2012, 卷号: 78, 期号: 2, 页码: 182-185
作者:  Huang SZ;  Zhang XJ;  Li XY;  Jiang HZ;  Ma QY;  Wang PC;  Liu YQ;  Hu JM;  Zheng YT;  Zhou J*;  Zhao YX*;  jzhou@mail.kib.ac.cn;  zhaoyx1011@163.com
Adobe PDF(113Kb)  |  收藏  |  浏览/下载:163/6  |  提交时间:2012/03/20
Daphne Acutiloba  Thymelaeceae  Anti-hiv Activity  Phenols  
Potent Anti-HIV Activities and Mechanisms of Action of a Pine Cone Extract from Pinus yunnanensis 期刊论文
MOLECULES, 2012, 卷号: 17, 期号: 6, 页码: 6916-6929
作者:  Zhang X;  Yang LM;  Liu GM;  Liu YJ;  Zheng CB;  Lv YJ;  Li HZ;  Zheng YT*;  zhengyt@mail.kiz.ac.cn
Adobe PDF(366Kb)  |  收藏  |  浏览/下载:141/4  |  提交时间:2012/09/04
Pinus Yunnanensis  Pine Cone  Anti-hiv Activity  Reverse Transcriptase  Fusion  
Synthesis and biological evaluation of novel dihydro-aryl/alkylsulfanyl-cyclohexylmethyl-oxopyrimidines (S-DACOs) as high active anti-HIV agents 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 卷号: 21, 期号: 2, 页码: 694-697
作者:  He YP*;  Long J;  Zhang SS;  Li C;  Lai CC;  Zhang CS;  Li DX;  Zhang DH;  Wang H;  Cai QQ;  Zheng YT*;  yphe@ynu.edu.cn;  zhengyt@mail.kiz.ac.cn
Adobe PDF(395Kb)  |  收藏  |  浏览/下载:1658/7  |  提交时间:2011/03/15
Nnrtis  S-dabos  S-dacos  Anti Hiv-1 Activity  
Synthesis and biological evaluation of naphthyl phenyl ethers (NPEs) as novel nonnucleoside HIV-1 reverse transcriptase inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 卷号: 19, 期号: 14, 页码: 4220-4226
作者:  Gu SX;  Zhang X;  Zheng YT;  Yang SQ;  Chen FE*;  He QQ;  Yang LM;  Ma XD;  rfchen@fudan.edu.cn
Adobe PDF(416Kb)  |  收藏  |  浏览/下载:55/1  |  提交时间:2016/08/30
Hiv-1 Reverse Transcriptase  Nnrtis  Npes  Sar  Anti-hiv Activity